Abstract: With the rapid evolution in the basic types of drugs and the continuous emergence of innovative formulations and new therapeutic approaches,the complexity and difficulty of teaching pharmacokinetics courses have also increased.This paper explores the challenges posed by the development of pharmacy to the teaching of pharmacokinetics and the potential solutions.By optimizing both the content and methods of instruction,the teaching team enhances the course's relevance and practical value,fosters students' interest,deepens their understanding and application of course knowledge,and broadens their perspectives and innovative thinking.These efforts are aimed at meeting the growing demands for talent in the evolving medical and pharmaceutical industry.